SCHEMBL19416975

SCHEMBL19416975

N#Cc1cnc(C2(F)CCNCC2)c(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
GRM5 P41594 3/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
MAPKAPK2 P49137 1/20 0.33
CHEK1 O14757 1/20 0.32
ALDH1A1 P00352 1/20 0.31
USP2 O75604 1/20 0.31
APP P05067 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16000814 0.87 HTT (0.36) HTTGRM5APPBACE1BACE2
SCHEMBL19416995 0.74 CYP2D6 (0.37)
SCHEMBL17644320 0.73 TRPV1 (0.39) CHRNB2CHRNA4ALDH1A1
SCHEMBL4289160 0.71 TRPV1 (0.52)
SCHEMBL3624558 0.71 TRPV1 (0.52)
SCHEMBL12686755 0.71 MAPKAPK2 (0.39) MAPKAPK2ALDH1A1USP2
SCHEMBL15035158 0.70 TRPV1 (0.41)
SCHEMBL14935719 0.70 TRPV1 (0.49)
SCHEMBL12073070 0.70 TRPV1 (0.54)
SCHEMBL12073818 0.70 TRPV1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709609-B1 HETEROCYCLIC COMPOUNDS SHIONOGI & CO (JP) 2017-10-04 EP disclosed