SCHEMBL19418016

SCHEMBL19418016

Cc1c(O)cc(O)c2c1CC(=O)/C=C/CC/C=C/CCOC2=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.51
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
MAPT P10636 3/20 0.33
HSP90AA1 P07900 2/20 0.33
GAA P10253 2/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NLRP3 Q96P20 1/20 0.33
CBR1 P16152 1/20 0.33
PTGS2 P35354 1/20 0.33
ACLY P53396 1/20 0.33
FTO Q9C0B1 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10150174 0.85 HSP90AB1 (0.66) HSP90AB1MAOAMAOBF13A1TGM2
SCHEMBL19418509 0.82 HSP90AB1 (0.47) HSP90AB1MAOAMAOBF13A1TGM2
SCHEMBL10150456 0.81 HSP90AB1 (0.78) HSP90AB1MAOAMAOBF13A1TGM2
SCHEMBL13080872 0.80 HSP90AB1 (0.35) HSP90AB1MAOAMAOB
SCHEMBL14293707 0.78 HSP90AB1 (0.58) HSP90AB1MAOAMAOBF13A1TGM2
SCHEMBL10150176 0.76 F13A1 (0.58) HSP90AB1F13A1TGM2MAPTHSP90AA1
SCHEMBL10150827 0.74 HSP90AB1 (0.46) HSP90AB1MAOAMAOBF13A1TGM2
SCHEMBL12384130 0.73 RAB9A (0.35) MAPTRAB9AHPGDSMN1; SMN2
SCHEMBL12423844 0.73 RAB9A (0.35) MAPTRAB9AHPGDSMN1; SMN2
SCHEMBL15702282 0.73 RAB9A (0.35) MAPTRAB9AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed