SCHEMBL19418239

SCHEMBL19418239

N=C1/C=C/CC/C=C/CCOC(=O)c2c(CO)cc(O)c(Cl)c2C1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 3/20 0.41
HSP90AA1 P07900 1/20 0.32
STAT6 P42226 1/20 0.30
SMAD3 P84022 1/20 0.30
SMAD2 Q15796 1/20 0.30
ACLY P53396 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10186746 0.89 HSP90AB1 (0.52) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL19418327 0.89 HSP90AB1 (0.52) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL19418380 0.85 HSP90AB1 (0.44) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL20840851 0.82 HSP90AB1 (0.50) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL10150174 0.76 HSP90AB1 (0.66) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL18871691 0.75 HSP90AB1 (0.44) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL20840838 0.74 HSP90AB1 (0.48) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL19418461 0.74 HSP90AB1 (0.52) HSP90AB1HSP90AA1STAT6SMAD3SMAD2
SCHEMBL17787723 0.74 F13A1 (0.45) HSP90AB1HSP90AA1
SCHEMBL20840837 0.73 HSP90AB1 (0.42) HSP90AB1HSP90AA1STAT6SMAD3SMAD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed