SCHEMBL19418404

SCHEMBL19418404

CC1CC2OC2CC/C=C/C(=O)Cc2cc(O)cc(N)c2C(=O)O1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 4/20 0.63
F13A1 P00488 1/20 0.57
TGM2 P21980 1/20 0.57
MKNK2 Q9HBH9 5/20 0.40
MAPT P10636 3/20 0.40
HSP90AA1 P07900 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
RAB9A P51151 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CBR1 P16152 2/20 0.40
GAA P10253 2/20 0.40
NLRP3 Q96P20 1/20 0.40
GEMIN4 P57678 1/20 0.40
HSF1 Q00613 1/20 0.40
PTGS2 P35354 1/20 0.40
ACLY P53396 1/20 0.40
FTO Q9C0B1 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monocillin Iii SCHEMBL10150121 0.90 HSP90AB1 (0.71) HSP90AB1F13A1TGM2MKNK2MAPT
Monocillin Iii SCHEMBL10150122 0.90 HSP90AB1 (0.71) HSP90AB1F13A1TGM2MKNK2MAPT
Monocillin Iii SCHEMBL10150575 0.90 HSP90AB1 (0.71) HSP90AB1F13A1TGM2MKNK2MAPT
SCHEMBL19418488 0.83 HSP90AB1 (0.61) HSP90AB1F13A1TGM2MKNK2MAPT
Pochonin A SCHEMBL10150715 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1
Pochonin A SCHEMBL10150818 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1
Pochonin A SCHEMBL10150114 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1
Pochonin A SCHEMBL10150819 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1
Pochonin A SCHEMBL19418057 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1
Pochonin A SCHEMBL10150463 0.78 HSP90AB1 (1.00) HSP90AB1F13A1TGM2MAPTHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed