SCHEMBL19418488

SCHEMBL19418488

C[C@H]1C/C=C/CC/C=C/C(=O)Cc2cc(O)cc(N)c2C(=O)O1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.61
F13A1 P00488 1/20 0.60
TGM2 P21980 1/20 0.60
MKNK2 Q9HBH9 6/20 0.54
FLT3 P36888 6/20 0.44
KIT P10721 6/20 0.44
PDGFRA P16234 6/20 0.44
KDR P35968 6/20 0.44
FLT4 P35916 4/20 0.44
FLT1 P17948 3/20 0.44
PDGFRB P09619 3/20 0.44
MAP2K1 Q02750 3/20 0.44
CCNA2 P20248 4/20 0.43
CDK2 P24941 4/20 0.43
CCNA1 P78396 4/20 0.43
MKNK1 Q9BUB5 3/20 0.43
PLK4 O00444 2/20 0.43
CDK1 P06493 2/20 0.43
AXL P30530 2/20 0.43
CDK5 Q00535 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10150507 0.88 F13A1 (0.77) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150038 0.88 F13A1 (0.77) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150437 0.88 F13A1 (0.77) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL14293730 0.87 HSP90AB1 (0.62) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL19418404 0.83 HSP90AB1 (0.63) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150144 0.80 KDR (0.67) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150367 0.77 HSP90AB1 (0.56) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150430 0.77 HSP90AB1 (0.56) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL10150199 0.77 HSP90AB1 (0.56) HSP90AB1F13A1TGM2MKNK2FLT3
SCHEMBL4510614 0.77 MKNK2 (0.63) HSP90AB1F13A1TGM2MKNK2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136799-B1 MACROCYCLIC COMPOUNDS USEFUL AS INHIBITORS OF KINASES AND HSP90 UNIV STRASBOURG (FR) 2017-10-04 EP disclosed