SCHEMBL194499

SCHEMBL194499

CCN(CC)c1ccc(C=C2SC(=S)NC2=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 3/20 1.00
CRHR2 Q13324 3/20 1.00
MYC P01106 3/20 0.68
MAX P61244 3/20 0.68
NPC1 O15118 1/20 0.68
RAB9A P51151 1/20 0.68
GSK3B P49841 1/20 0.67
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
POLB P06746 1/20 0.65
GPR35 Q9HC97 1/20 0.65
NAT1 P18440 5/20 0.61
CISD1 Q9NZ45 1/20 0.61
KDM4E B2RXH2 1/20 0.60
ALDH1A1 P00352 1/20 0.60
LMNA P02545 1/20 0.60
GAA P10253 1/20 0.60
MAPT P10636 1/20 0.60
MAPK1 P28482 1/20 0.60
NTSR1 P30989 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1249353 1.00 CRHBP (1.00) CRHBPCRHR2MYCMAXNPC1
SCHEMBL194498 1.00 CRHBP (1.00) CRHBPCRHR2MYCMAXNPC1
SCHEMBL14891689 0.95 CRHBP (0.90) CRHBPCRHR2MYCMAXNPC1
SCHEMBL14891688 0.95 CRHBP (0.90) CRHBPCRHR2MYCMAXNPC1
SCHEMBL12218499 0.89 CRHBP (0.81) CRHBPCRHR2MYCMAXNPC1
SCHEMBL4101541 0.88 CRHBP (0.79) CRHBPCRHR2NPC1RAB9AGSK3B
SCHEMBL4101538 0.88 CRHBP (0.79) CRHBPCRHR2NPC1RAB9AGSK3B
SCHEMBL8177383 0.85 CRHBP (0.74) CRHBPCRHR2MYCMAXNPC1
SCHEMBL4100036 0.84 CRHBP (0.73) CRHBPCRHR2NPC1RAB9AGSK3B
SCHEMBL4100041 0.84 CRHBP (0.73) CRHBPCRHR2NPC1RAB9AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 248 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11382868-B2 Transdermal UV-curable hydrogel resin, hydrogel curing the same and cataplasm containing the same ICURE PHARMACEUTICAL INC. (KR) 2022-07-12 US claimed
US-20190046463-A1 ULTRAVIOLET-HARDENING HYDROGEL RESIN AND HYDROGEL FOR TRANSDERMAL ADMINISTRATION, AND CATAPLASM AGENT CONTAINING SAME ICURE PHARMACEUTICAL INC. (KR) 2019-02-14 US claimed
EP-3415141-A1 ULTRAVIOLET-HARDENING HYDROGEL RESIN AND HYDROGEL FOR TRANSDERMAL ADMINISTRATION, AND CATAPLASM AGENT CONTAINING SAME Icure Pharmaceutical Inc. (KR) 2018-12-19 EP claimed
EP-0527186-A4 UNIV ILLINOIS (US) 1995-01-18 EP claimed
EP-0527186-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS The Board of Trustees for the University of Illinois (US) 1993-02-17 EP claimed
WO-1991016820-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1991-11-14 WO claimed
JP-54133880-A None JP disclosed
EP-4743828-A1 PHOTOCURABLE AS WELL AS THERMALLY CURABLE COMPOSITIONS SUITABLE FOR LOW TEMPERATURE CURING BASF SE (DE) 2026-05-20 EP disclosed
US-20250149336-A1 PHOTORESIST COMPOSITION AND METHOD OF MANUFACTURING INTEGRATED CIRCUIT DEVICE USING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2025-05-08 US disclosed
CN-114129544-B Ultraviolet curable hydrogel resin for transdermal administration, hydrogel, and cataplasm comprising same Icure药品株式会社 2025-03-21 CN disclosed
CN-119403840-A Photocurable composition, method for producing cured film, solid-state imaging element, image display device, and radical polymerization initiator 富士胶片株式会社 2025-02-07 CN disclosed
WO-2025011754-A1 PHOTOCURABLE AS WELL AS THERMALLY CURABLE COMPOSITIONS SUITABLE FOR LOW TEMPERATURE CURING BASF SE (DE) 2025-01-16 WO disclosed
EP-4114825-B1 OXIME ESTER PHOTOINITIATORS BASF SE (DE) 2024-11-20 EP disclosed
EP-0733649-A1 Peroxycarboxylic ester initiators derived from nitrogen heterocycles MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-09-25 EP disclosed
US-5527921-A USEFUL IN PHOTOPOLYMERIZABLE COMPOSITIONS AND PHOTOSENSITIVE ELEMENTS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-06-18 US disclosed
EP-0527186-A4 UNIV ILLINOIS (US) 1995-01-18 EP disclosed
US-5242892-A With 5-aminolevulinic acid THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1993-09-07 US disclosed
EP-0527186-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS The Board of Trustees for the University of Illinois (US) 1993-02-17 EP disclosed
WO-1991016820-A1 PHOTODYNAMIC PLANT DEFOLIANTS AND CHLOROPHYLL BIOSYNTHESIS MODULATORS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 1991-11-14 WO disclosed
JP-S54133880-A ETCHING METHOD HITACHI LTD 1979-10-17 JP disclosed