SCHEMBL19488602

SCHEMBL19488602

C=C1CCN[C@@H]1c1nc2ccc(C#Cc3ccc(-c4cnc([C@@H]5CCCN5)[nH]4)cc3)cc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.42
DGAT1 O75907 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SSTR3 P32745 1/20 0.31
NPY5R Q15761 1/20 0.30
ADORA2A P29274 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16572630 0.90 SCN10A (0.51) SCN10ADGAT1NPC1RAB9ASSTR3
SCHEMBL16405116 0.90 SCN10A (0.51) SCN10ADGAT1NPC1RAB9ASSTR3
SCHEMBL10144768 0.90 SCN10A (0.51) SCN10ADGAT1NPC1RAB9ASSTR3
SCHEMBL19488818 0.87 SCN10A (0.41) SCN10ANPY5R
SCHEMBL19488496 0.81 SCN10A (0.43) SCN10ANPC1RAB9A
SCHEMBL19488796 0.80 SCN10A (0.45) SCN10ANPC1RAB9ANPY5R
SCHEMBL882760 0.80 MAPK13 (0.41) SCN10ASSTR3NPY5RKCNH2
SCHEMBL15388617 0.79 SCN10A (0.45) SCN10ADGAT1NPC1RAB9ANPY5R
SCHEMBL15388620 0.79 SCN10A (0.45) SCN10ADGAT1NPC1RAB9ANPY5R
SCHEMBL13192596 0.79 SCN10A (0.56) SCN10ANPC1RAB9ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601188-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-10-18 EP disclosed