SCHEMBL19491900

SCHEMBL19491900

COc1cc(N2CCN([S+](C)[O-])CC2)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.44
ALDH1A1 P00352 6/20 0.43
LMNA P02545 2/20 0.43
CYP3A4 P08684 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 3/20 0.42
GAA P10253 3/20 0.42
MAPT P10636 3/20 0.42
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
RECQL P46063 1/20 0.42
PTK2B Q14289 1/20 0.42
RAD52 P43351 1/20 0.39
HTR1A P08908 1/20 0.39
HTR7 P34969 1/20 0.39
CHEK1 O14757 1/20 0.39
MEN1 O00255 1/20 0.37
S100B P04271 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15358736 0.87 ALDH1A1 (0.53) SIRT6ALDH1A1LMNACYP3A4TDP1
SCHEMBL29446146 0.81 MAPT (0.63) SIRT6ALDH1A1CYP3A4TDP1TSHR
SCHEMBL438444 0.81 MAPT (0.63) SIRT6ALDH1A1CYP3A4TDP1TSHR
SCHEMBL2974453 0.81 ALDH1A1 (0.59) ALDH1A1LMNACYP3A4TDP1TSHR
SCHEMBL11291219 0.81 ALDH1A1 (0.43) SIRT6ALDH1A1LMNACYP3A4TDP1
SCHEMBL24900714 0.80 ALDH1A1 (0.46) SIRT6ALDH1A1LMNACYP3A4TDP1
Hydrochloric Acid SCHEMBL3504109 0.80 MAPT (0.61) SIRT6ALDH1A1CYP3A4TDP1TSHR
SCHEMBL2821837 0.80 MAPT (0.48) ALDH1A1LMNACYP3A4TDP1TSHR
SCHEMBL10128598 0.80 ALDH1A1 (0.59) ALDH1A1LMNACYP3A4TDP1TSHR
SCHEMBL30340649 0.80 ALDH1A1 (0.59) ALDH1A1LMNACYP3A4TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3293183-B1 INHIBITOR COMPOUNDS CANCER RESEARCH TECH LTD (GB) 2019-07-24 EP disclosed
EP-3293183-A1 INHIBITOR COMPOUNDS Cancer Research Technology Ltd. (GB) 2018-03-14 EP disclosed
EP-2892889-B1 INHIBITOR COMPOUNDS CANCER RES TECH LTD (GB) 2017-10-18 EP disclosed