SCHEMBL19503550

SCHEMBL19503550

CNc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IKZF2 Q9UKS7 10/20 0.74
CRBN Q96SW2 10/20 0.72
CSNK1A1 P48729 2/20 0.67
IKZF1 Q13422 1/20 0.57
GSPT1 P15170 1/20 0.56
DDB1 Q16531 1/20 0.56
IKZF3 Q9UKT9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25571538 1.00 IKZF2 (0.74) IKZF2CRBNCSNK1A1IKZF1GSPT1
SCHEMBL29547357 1.00 IKZF2 (0.74) IKZF2CRBNCSNK1A1IKZF1GSPT1
SCHEMBL19503631 0.91 CRBN (0.69) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL23226142 0.89 CRBN (0.70) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL31546799 0.88 CRBN (0.72) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL23729630 0.88 CRBN (0.72) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL19503565 0.87 IKZF2 (0.73) IKZF2CRBNCSNK1A1DDB1
SCHEMBL24637334 0.87 CRBN (0.71) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL25628768 0.87 CRBN (0.74) IKZF2CRBNCSNK1A1GSPT1DDB1
SCHEMBL23535299 0.86 CRBN (0.74) IKZF2CRBNCSNK1A1GSPT1DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12559486-B2 Tau-protein targeting compounds and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-02-24 US disclosed
US-20240217962-A1 TAU-PROTEIN TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. 2024-07-04 US disclosed
US-11912699-B2 Tau-protein targeting compounds and associated ARVINAS OPERATIONS, INC. (US) 2024-02-27 US disclosed
US-11912699-B2 Tau-protein targeting compounds and associated ARVINAS OPERATIONS, INC. (US) 2024-02-27 US disclosed
US-11912699-B2 Tau-protein targeting compounds and associated ARVINAS OPERATIONS, INC. (US) 2024-02-27 US disclosed
WO-2024006881-A1 WEE1 DEGRADING COMPOUNDS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2024-01-04 WO disclosed
WO-2024006403-A2 SELECTIVE HISTONE DEACETYLASE 8 (HDAC8) DEGRADERS AND METHODS OF USE THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-01-04 WO disclosed
US-11833142-B2 3-(5-amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof NOVARTIS AG (CH) 2023-12-05 US disclosed
WO-2023220722-A2 PAK1 DEGRADERS AND METHODS OF USE THEREOF INSTITUTE FOR CANCER RESEARCH D/B/A THE RESEARCH INSTITUTE OF FOX CHASE CANCER CENTER (US) 2023-11-16 WO disclosed
EP-3820574-B1 3-(5-AMINO-1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF IKAROS FAMILY ZINC FINGER 2 (IKZF2)-DEPENDENT DISEASES NOVARTIS AG (CH) 2023-08-09 EP disclosed
WO-2021242982-A1 GALECTIN-3 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-12-02 WO disclosed
WO-2021222542-A1 5-AMINO-2-PIPERIDINON-3-YL-1-OXOISOINDOLINE DERIVATIVES FOR DEGRADATION OF IKZF2 DEGRADERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2021-11-04 WO disclosed
WO-2021078301-A1 PROTEIN DEGRADING AGENT AND USE THEREOF IN TREATMENT OF DISEASES 上海科技大学 2021-04-29 WO disclosed
WO-2021068380-A1 PREPARATION OF DEGRADATION COMPOUND TARGETING BTK PROTEIN, AND APPLICATION THEREOF IN TREATING AUTOIMMUNE DISEASES AND TUMORS 清华大学 2021-04-15 WO disclosed
WO-2020227325-A1 HETEROBIFUNCTIONAL COMPOUNDS AS DEGRADERS OF HPK1 ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2020-11-12 WO disclosed
WO-2020081880-A1 COMPOSITIONS TARGETING SENESCENT CELLS AND THE USES THEREOF BIOVENTURES, LLC (US) 2020-04-23 WO disclosed
WO-2020038415-A1 TROPOMYOSIN RECEPTOR KINASE (TRK) DEGRADATION COMPOUNDS AND METHODS OF USE CULLGEN (SHANGHAI), INC. (CN) 2020-02-27 WO disclosed
WO-2019173516-A1 SERINE THREONINE KINASE (AKT) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2019-09-12 WO disclosed
WO-2019165189-A1 PROTEIN ARGININE METHYLTRANSFERASE 5 (PRMT5) DEGRADATION / DISRUPTION COMPOUNDS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2019-08-29 WO disclosed
WO-2017184995-A1 COMPOUNDS THAT INDUCE DEGRADATION OF ANTI-APOPTOTIC BCL-2 FAMILY PROTEINS AND THE USES THEREOF BIOVENTURES, LLC (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11912699-B2 Tau-protein targeting compounds and associated MAPT, VHL, CRBN IKZF2 3079/4885CRBN 3/4885CSNK1A1 868/4885
US-20240217962-A1 TAU-PROTEIN TARGETING COMPOUNDS AND ASSOCIATED METHODS OF USE VHL, CRBN, MAPT IKZF2 3413/4885CRBN 2/4885CSNK1A1 829/4885
US-11833142-B2 3-(5-amino-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof RXFP3, RXFP1, NPY2R IKZF2 3369/4885CRBN 3123/4885CSNK1A1 486/4885
US-12559486-B2 Tau-protein targeting compounds and associated methods of use UBQLN2, UBQLN1, CRBN IKZF2 3718/4885CRBN 3/4885CSNK1A1 281/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.