SCHEMBL19503565

SCHEMBL19503565

CC(C)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IKZF2 Q9UKS7 10/20 0.73
CRBN Q96SW2 10/20 0.68
DDB1 Q16531 1/20 0.67
CSNK1A1 P48729 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19503714 0.91 CRBN (0.67) IKZF2CRBNDDB1CSNK1A1
SCHEMBL25571538 0.87 IKZF2 (0.74) IKZF2CRBNDDB1CSNK1A1
SCHEMBL19503550 0.87 IKZF2 (0.74) IKZF2CRBNDDB1CSNK1A1
SCHEMBL29547357 0.87 IKZF2 (0.74) IKZF2CRBNDDB1CSNK1A1
SCHEMBL23226142 0.86 CRBN (0.70) IKZF2CRBNDDB1CSNK1A1
SCHEMBL23535299 0.86 CRBN (0.74) IKZF2CRBNDDB1CSNK1A1
SCHEMBL23729630 0.85 CRBN (0.72) IKZF2CRBNDDB1CSNK1A1
SCHEMBL31546799 0.85 CRBN (0.72) IKZF2CRBNDDB1CSNK1A1
SCHEMBL24062315 0.85 IKZF2 (1.00) IKZF2CRBNDDB1CSNK1A1
SCHEMBL21617629 0.85 IKZF2 (1.00) IKZF2CRBNDDB1CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230210999-A1 TARGETED PROTEASE DEGRADATION (TED) PLATFORM EUBULUS BIOTHERAPEUTICS (HONG KONG) LIMITED (HK) 2023-07-06 US disclosed
US-20220313829-A1 EGFR PROTEIN DEGRADANT AND ANTI-TUMOR APPLICATION THEREOF SHANGHAITECH UNIVERSITY (CN) 2022-10-06 US disclosed
US-11319316-B2 Compounds that induce degradation of anti-apoptotic Bcl-2 family proteins and the uses thereof BIOVENTURES, LLC (US) 2022-05-03 US disclosed
US-20200331905-A1 Compounds That Induce Degradation of Anti-Apoptotic BCL-2 Family Proteins and the Uses Thereof BIOVENTURES, LLC 2020-10-22 US disclosed
US-10807977-B2 Compounds that induce degradation of anti-apoptotic Bcl-2 family proteins and the uses thereof BIOVENTURES, LLC (US) 2020-10-20 US disclosed
WO-2020081880-A1 COMPOSITIONS TARGETING SENESCENT CELLS AND THE USES THEREOF BIOVENTURES, LLC (US) 2020-04-23 WO disclosed
US-20190135801-A1 COMPOUNDS THAT INDUCE DEGRADATION OF ANTI-APOPTOTIC BCL-2 FAMILY PROTEINS AND THE USES THEREOF BIOVENTURES, LLC 2019-05-09 US disclosed
US-20190054097-A1 COMPOSITIONS TARGETING SENESCENT CELLS AND THE USES THEREOF BIOVENTURES, LLC 2019-02-21 US disclosed
WO-2017184995-A1 COMPOUNDS THAT INDUCE DEGRADATION OF ANTI-APOPTOTIC BCL-2 FAMILY PROTEINS AND THE USES THEREOF BIOVENTURES, LLC (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230210999-A1 TARGETED PROTEASE DEGRADATION (TED) PLATFORM UCHL3, UBE2L3, ADAM33 IKZF2 2378/4885CRBN 286/4885DDB1 1415/4885
US-20200331905-A1 Compounds That Induce Degradation of Anti-Apoptotic BCL-2 Family Proteins and the Uses Thereof BCL2, BAX, BCL2L1 IKZF2 556/4885CRBN 520/4885DDB1 134/4885
US-20220313829-A1 EGFR PROTEIN DEGRADANT AND ANTI-TUMOR APPLICATION THEREOF EGFR, ERBB2, ERBB3 IKZF2 3455/4885CRBN 3528/4885DDB1 1479/4885
US-20190135801-A1 COMPOUNDS THAT INDUCE DEGRADATION OF ANTI-APOPTOTIC BCL-2 FAMILY PROTEINS AND THE USES THEREOF BCL2, BAX, BCL2L1 IKZF2 556/4885CRBN 520/4885DDB1 134/4885
US-11319316-B2 Compounds that induce degradation of anti-apoptotic Bcl-2 family proteins and the uses thereof BCL2, BAX, BCL2L1 IKZF2 556/4885CRBN 520/4885DDB1 134/4885
US-10807977-B2 Compounds that induce degradation of anti-apoptotic Bcl-2 family proteins and the uses thereof BCL2, BAX, BCL2L1 IKZF2 556/4885CRBN 520/4885DDB1 134/4885
US-20190054097-A1 COMPOSITIONS TARGETING SENESCENT CELLS AND THE USES THEREOF TP53, MCL1, LIMS1 IKZF2 1680/4885CRBN 1187/4885DDB1 55/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.