SCHEMBL19554199

SCHEMBL19554199

Cc1csc2ccc(C(=O)Nc3ccc(Cl)cc3C(=O)O)cc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 11/20 0.57
AKR1C4 P17516 1/20 0.55
AKR1C3 P42330 1/20 0.55
AKR1C2 P52895 1/20 0.55
AKR1C1 Q04828 1/20 0.55
CA2 P00918 3/20 0.54
CA9 Q16790 3/20 0.54
CA12 O43570 2/20 0.54
CA1 P00915 2/20 0.54
CA7 P43166 1/20 0.54
CYP2A6 P11509 1/20 0.51
KCNK2 O95069 1/20 0.50
KCNK10 P57789 1/20 0.50
KDM4E B2RXH2 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6353448 0.78 SERPINE1 (0.64) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL19554217 0.78 SERPINE1 (0.58) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL19554265 0.75 SERPINE1 (0.58) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL19554134 0.75 SERPINE1 (0.68) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL17842775 0.74 CYP2A6 (0.53) CA2CA9CA12CA1CA7
SCHEMBL6358123 0.73 SERPINE1 (0.89) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL6349535 0.73 SERPINE1 (0.74) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL6351321 0.73 SERPINE1 (0.89) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL420142 0.73 SERPINE1 (1.00) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11231268 0.72 CHEK1 (0.70) SERPINE1AKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO claimed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed