SCHEMBL19583155

SCHEMBL19583155

CN(CC#Cc1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.57
PPARG P37231 1/20 0.55
PYCR1 P32322 1/20 0.50
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
THPO P40225 1/20 0.47
EGLN1 Q9GZT9 1/20 0.46
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
HTR2A P28223 1/20 0.44
CYP2A6 P11509 1/20 0.43
NPSR1 Q6W5P4 2/20 0.43
APP P05067 1/20 0.42
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136691 0.81 CYP2A6 (0.61) GRM5PYCR1CYP3A4CYP2C9CYP2C19
SCHEMBL8331122 0.81 GRM5 (0.53) GRM5PPARGPYCR1CYP3A4CYP1A2
SCHEMBL22485593 0.79 GRM5 (0.51) GRM5PPARGPYCR1CYP3A4EGLN1
SCHEMBL14269510 0.76 GRM5 (0.49) GRM5PPARGEGLN1MEN1ALDH1A1
SCHEMBL46288 0.73 KCNH2 (0.58) PYCR1CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL19420119 0.73 PYCR1 (0.47) PYCR1CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL5703380 0.73 GRM5 (1.00) GRM5CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL304704 0.72 MAOB (0.47) GRM5PPARGPYCR1CYP3A4NPSR1
SCHEMBL6929485 0.72 CA12 (0.47) GRM5PPARGPYCR1CYP3A4MEN1
SCHEMBL5982497 0.72 MAOB (0.53) GRM5PYCR1CYP3A4CYP1A2BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111875552-B Amino-substituted 1,2, 3-triazole compound and synthesis method and application thereof 海南师范大学 2022-06-21 CN disclosed
CN-111875552-A Amino-substituted 1,2, 3-triazole compound and synthesis method and application thereof 海南师范大学 2020-11-03 CN disclosed
US-10112189-B2 Trans-metallated MOF catalyst KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2018-10-30 US disclosed
US-20180280949-A1 TRANS-METALLATED MOF CATALYST KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2018-10-04 US disclosed
US-9975114-B2 Metal organic frameworks as catalysts and hydrocarbon oxidation methods thereof KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2018-05-22 US disclosed
US-20170326536-A1 METAL ORGANIC FRAMEWORKS AS CATALYSTS AND HYDROCARBON OXIDATION METHODS THEREOF KING FAHD UNIVERSITY OF PETROLEUM AND MINERALS (SA) 2017-11-16 US disclosed