SCHEMBL19595173

SCHEMBL19595173

CCC1NC(=O)CNC(=O)C(CCCNC(=N)N)NC(=O)C(C(C)C)N(C)C(=O)C(Cc2ccccc2)NC1=O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.49
ITGAV P06756 6/20 0.49
ITGB5 P18084 4/20 0.49
ITGA2B P08514 1/20 0.49
ITGB6 P18564 1/20 0.49
CXCR4 P61073 1/20 0.47
MC4R P32245 10/20 0.46
MC5R P33032 10/20 0.46
MC3R P41968 10/20 0.46
MC1R Q01726 10/20 0.46
ITGB1 P05556 1/20 0.45
ITGA5 P08648 1/20 0.45
KDM4A O75164 1/20 0.44
TSLP Q969D9 1/20 0.43
HDAC4 P56524 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12468724 0.94 ITGB3 (0.47) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL12467279 0.94 ITGB3 (0.49) ITGB3ITGAVITGB5ITGA2BITGB6
Cilengitide SCHEMBL22594705 0.93 ITGB3 (0.59) ITGB3ITGAVITGB5ITGA2BITGB6
Cilengitide SCHEMBL451423 0.93 ITGB3 (0.59) ITGB3ITGAVITGB5ITGA2BITGB6
Cilengitide SCHEMBL16920496 0.93 ITGB3 (0.59) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL16923811 0.91 ITGB3 (0.52) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL12016720 0.88 ITGB3 (0.46) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL24202406 0.86 ITGB3 (0.48) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL22807659 0.86 ITGB3 (0.48) ITGB3ITGAVITGB5ITGA2BITGB6
SCHEMBL16920494 0.86 ITGB3 (0.51) ITGB3ITGAVITGB5ITGA2BITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3243530-A1 INTEGRIN RECEPTOR ANTAGONISTS AND THEIR USE Allegro Pharmaceuticals, Inc. (US) 2017-11-15 EP disclosed