SCHEMBL19609239

SCHEMBL19609239

NCC(=O)N1CCc2sc(NC=O)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.39
F2 P00734 1/20 0.37
TPSAB1 Q15661 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
KDM1A O60341 5/20 0.36
PRMT5 O14744 2/20 0.34
WDR77 Q9BQA1 2/20 0.34
CHEK1 O14757 1/20 0.33
AOC3 Q16853 1/20 0.33
P2RX3 P56373 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086176 0.71 KDM1A (0.51) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL17544835 0.70 HDAC6 (0.42) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL19086200 0.69 HDAC6 (0.48) HDAC6KDM1APRMT5WDR77MEN1
SCHEMBL28956427 0.65 HDAC6 (0.41) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL19086224 0.65 HDAC6 (0.42) HDAC6KDM1AMEN1KMT2ADPP8
SCHEMBL3441635 0.64 HDAC6 (0.43) HDAC6F2TPSAB1TPSD1TPSG1
Hydrochloric Acid SCHEMBL27170981 0.64 DPP8 (0.62) MEN1KMT2ADPP8DPP7KDM4E
SCHEMBL3555661 0.63 NOTUM (0.47) HDAC6F2TPSAB1TPSD1TPSG1
SCHEMBL19303081 0.62 ESR2 (0.52) HDAC6KDM4E
SCHEMBL2921885 0.62 MAPT (0.44) HDAC6F2TPSAB1TPSD1TPSG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017195216-A1 CYCLOPROPYL-AMIDE COMPOUNDS AS DUAL LSD1/HDAC INHIBITORS JUBILANT BIOSYS LIMITED (IN) 2017-11-16 WO disclosed