SCHEMBL1961097

SCHEMBL1961097

CNc1nc(SC)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 12/20 0.74
ADORA1 P30542 12/20 0.74
KDM4E B2RXH2 1/20 0.64
PKM P14618 1/20 0.64
ADORA2A P29274 5/20 0.63
ADORA2B P29275 5/20 0.63
HTR2A P28223 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
MAPK1 P28482 1/20 0.62
CYP2C19 P33261 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3692106 1.00 ADORA3 (0.74) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL28120773 0.92 KDM4E (0.64) ADORA3ADORA1KDM4EPKMADORA2A
Adenosine SCHEMBL28274972 0.91 ADORA3 (0.68) ADORA3ADORA1ADORA2AADORA2BMAPK1
SCHEMBL21685900 0.90 ADORA3 (0.61) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL8818470 0.88 KDM4E (0.59) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL28952609 0.88 KDM4E (0.59) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL8818497 0.88 KDM4E (0.59) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL29278767 0.87 ADORA3 (0.59) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL18171845 0.86 KDM4E (0.57) ADORA3ADORA1KDM4EPKMADORA2A
SCHEMBL18371513 0.86 KDM4E (0.57) ADORA3ADORA1KDM4EPKMADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2655 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4705468-A1 MAMMALIAN POLYCISTRONIC EXPRESSION SYSTEM FOR DIRECT TRANSLATION FROM RNA AND SECRETION OF CARGO California Institute of Technology (US) 2026-03-11 EP claimed
EP-4634380-A1 INTERNAL RIBOSOME ENTRY SITES FOR IMPROVED POLYNUCLEOTIDE TRANSLATION ModernaTX, Inc. (US) 2025-10-22 EP claimed
EP-4632075-A2 METHOD FOR REDUCING IMMUNOGENICITY OF RNA BioNTech SE (DE) 2025-10-15 EP claimed
US-20250304965-A1 DOUBLE-STRANDED RNA MOLECULE AND PHARMACEUTICAL USE THEREOF MACAU UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2025-10-02 US claimed
EP-4029522-B1 METHOD FOR REDUCING IMMUNOGENICITY OF RNA BioNTech SE (DE) 2025-08-13 EP claimed
WO-2025137275-A1 NOVEL CAS NUCLEASES AND POLYNUCLEOTIDES ENCODING THE SAME MODERNATX, INC. (US) 2025-06-26 WO claimed
EP-4565692-A2 INTERNAL RIBOSOME ENTRY SITES FOR IMPROVED POLYNUCLEOTIDE TRANSLATION ModernaTX, Inc. (US) 2025-06-11 EP claimed
US-20250019719-A1 Purification and Purity Assessment of RNA Molecules Synthesized with Modified Nucleosides THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2025-01-16 US claimed
CN-117866948-B Negative selection method and system for purifying circular nucleic acid 上海环码生物医药有限公司 2024-12-13 CN claimed
US-20240366793-A1 MAMMALIAN POLYCISTRONIC EXPRESSION SYSTEM FOR DIRECT TRANSLATION FROM RNA AND SECRETION OF CARGO CALIFORNIA INST OF TECHN (US) 2024-11-07 US claimed
EP-3656872-A1 LABEL-FREE ANALYSIS OF RNA CAPPING EFFICIENCY USING RNASE H, PROBES AND LIQUID CHROMATOGRAPHY/MASS SPECTROMETRY Novartis AG (CH) 2020-05-27 EP claimed
CN-110870871-A Methods and pharmaceutical compositions for treating cancer 澳门科技大学 2020-03-10 CN claimed
US-20200071695-A1 METHOD AND PHARMACEUTICAL COMPOSITION FOR TREATING CANCER INCREASEPHARM (HK) LIMITED (HK) 2020-03-05 US claimed
EP-3387150-B1 LABEL-FREE ANALYSIS OF RNA CAPPING EFFICIENCY USING RNASE H, PROBES AND LIQUID CHROMATOGRAPHY/MASS SPECTROMETRY NOVARTIS AG (CH) 2019-10-02 EP claimed
EP-3387150-A1 LABEL-FREE ANALYSIS OF RNA CAPPING EFFICIENCY USING RNASE H, PROBES AND LIQUID CHROMATOGRAPHY/MASS SPECTROMETRY Novartis AG (CH) 2018-10-17 EP claimed
US-9719084-B2 Co-transcriptional assembly of modified RNA nanoparticles THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2017-08-01 US claimed
WO-2017098468-A1 LABEL-FREE ANALYSIS OF RNA CAPPING EFFICIENCY USING RNASE H, PROBES AND LIQUID CHROMATOGRAPHY/MASS SPECTROMETRY NOVARTIS AG (CH) 2017-06-15 WO claimed
US-20150203842-A1 CO-TRANSCRIPTIONAL ASSEMBLY OF MODIFIED RNA NANOPARTICLES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES 2015-07-23 US claimed
WO-2014039809-A2 CO-TRANSCRIPTIONAL ASSEMBLY OF MODIFIED RNA NANOPARTICLES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2014-03-13 WO claimed
EP-2578685-A2 RNA containing modified nucleosides and methods of use thereof The Trustees of The University of Pennsylvania (US) 2013-04-10 EP claimed