SCHEMBL19617992

SCHEMBL19617992

COc1ccc(-c2nc3c(C)cccn3c2C(C)C)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.42
MTOR P42345 2/20 0.41
GAA P10253 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
ATM Q13315 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KDR P35968 1/20 0.40
MAPT P10636 3/20 0.39
CYP2A6 P11509 1/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18294576 0.85 CYP11B1 (0.50) JAK2MTORGAANPSR1KDM4E
SCHEMBL18293595 0.85 GAA (0.44) GAANPSR1KDM4ENPC1ALDH1A1
SCHEMBL18294600 0.83 GAA (0.61) JAK2MTORGAANPSR1KDM4E
Hydrochloric Acid SCHEMBL15716897 0.82 GAA (0.60) JAK2MTORGAANPSR1KDM4E
SCHEMBL15729914 0.81 JAK2 (0.42) JAK2MTORGAANPSR1KDM4E
SCHEMBL18293602 0.78 GAA (0.64) GAANPSR1KDM4ENPC1ALDH1A1
SCHEMBL22146345 0.70 ALDH1A1 (0.47) GAANPSR1KDM4ENPC1ALDH1A1
SCHEMBL14810539 0.69 CYP11B1 (0.55) GAANPSR1KDM4ENPC1ALDH1A1
SCHEMBL13561321 0.69 CYP2A6 (0.46) JAK2MTORCYP2A6PIK3CAHSD17B1
SCHEMBL10094701 0.68 CYP2A6 (0.57) MTORKDM4EALDH1A1HPGDCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9822118-B2 Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors ARRAY BIOPHARMA INC. (US) 2017-11-21 US disclosed