SCHEMBL19620247

SCHEMBL19620247

N=C(/C(COc1ccc(C2(O)CN(c3cncc(C(=O)O)c3)C2)c(Cl)c1)=C(\O)C1CC1)c1c(Cl)cccc1Cl

nearest known ligand 0.58

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.58
HSD17B13 Q7Z5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18724807 0.91 NR1H4 (0.55) NR1H4HSD17B13
SCHEMBL19725197 0.87 NR1H4 (0.60) NR1H4HSD17B13
SCHEMBL19738335 0.84 NR1H4 (0.58) NR1H4HSD17B13
SCHEMBL24357886 0.84 NR1H4 (0.49) NR1H4HSD17B13
SCHEMBL20749532 0.83 NR1H4 (0.52) NR1H4HSD17B13
SCHEMBL19725196 0.81 NR1H4 (0.58) NR1H4HSD17B13
SCHEMBL20749534 0.81 NR1H4 (0.46) NR1H4HSD17B13
SCHEMBL23773972 0.80 NR1H4 (0.38) NR1H4HSD17B13
SCHEMBL19738535 0.80 NR1H4 (0.61) NR1H4HSD17B13
SCHEMBL19620260 0.80 NR1H4 (0.55) NR1H4HSD17B13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246070-A1 NOVEL FXR (NR1H4) BINDING AND ACTIVITY MODULATING AZOLES Gilead Sciences, Inc. (US) 2017-11-22 EP disclosed