SCHEMBL19620248

SCHEMBL19620248

COC(=O)c1cccc([C@H]2C[C@](O)(c3ccc(OCC4C(c5c(Cl)cccc5Cl)=NOC4C4CC4)cc3Cl)C2)c1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.51
HSD17B13 Q7Z5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18724828 0.87 NR1H4 (0.59) NR1H4HSD17B13
SCHEMBL12879066 0.79 NR1H4 (0.51) NR1H4
SCHEMBL12879009 0.79 NR1H4 (0.48) NR1H4
SCHEMBL14562396 0.76 NR1H4 (0.85) NR1H4HSD17B13
SCHEMBL14605490 0.76 NR1H4 (0.85) NR1H4HSD17B13
SCHEMBL15929532 0.76 NR1H4 (0.85) NR1H4HSD17B13
SCHEMBL12879085 0.76 NR1H4 (0.58) NR1H4
SCHEMBL19230732 0.75 NR1H4 (0.34) NR1H4
SCHEMBL19202526 0.74 NR1H4 (0.64) NR1H4HSD17B13
SCHEMBL12879061 0.74 NR1H4 (0.49) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246070-A1 NOVEL FXR (NR1H4) BINDING AND ACTIVITY MODULATING AZOLES Gilead Sciences, Inc. (US) 2017-11-22 EP disclosed