SCHEMBL19622262

SCHEMBL19622262

N#Cc1ccc(Oc2ccc(P)c(CO)c2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.40
KCNH2 Q12809 2/20 0.40
SLC6A4 P31645 1/20 0.40
AR P10275 4/20 0.39
EPAS1 Q99814 3/20 0.38
SLC22A12 Q96S37 3/20 0.35
USP30 Q70CQ3 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
SLC22A11 Q9NSA0 1/20 0.35
FFAR1 O14842 2/20 0.34
TBXA2R P21731 1/20 0.34
SCN9A Q15858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29581919 0.75 AR (0.46) AREPAS1SLC22A12USP30
SCHEMBL29851244 0.75 AR (0.48) ARUSP30TBXA2R
SCHEMBL8616842 0.75 AR (0.48) ARUSP30TBXA2R
SCHEMBL8544623 0.74 AR (0.54) HTR2AKCNH2SLC6A4AREPAS1
SCHEMBL2989414 0.73 SLC6A4 (0.38) KCNH2SLC6A4AREPAS1SLC22A12
SCHEMBL8754808 0.72 AR (0.49) HTR2AKCNH2SLC6A4ARTBXA2R
SCHEMBL8616839 0.72 AR (0.48) HTR2AKCNH2SLC6A4ARSLC22A12
SCHEMBL29255047 0.72 AR (0.48) HTR2AKCNH2SLC6A4ARSLC22A12
SCHEMBL28671160 0.72 AR (0.48) HTR2AKCNH2SLC6A4ARSLC22A12
SCHEMBL9644087 0.72 AR (0.59) HTR2AKCNH2SLC6A4ARSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed