SCHEMBL19622265

SCHEMBL19622265

N#Cc1ccc(Oc2ccc3c(c2)COB3)c(OCC(=O)C=O)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.36
PPARD Q03181 3/20 0.36
PPARA Q07869 3/20 0.36
PDE4B Q07343 3/20 0.35
CHRM1 P11229 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
PDE1A P54750 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE7A Q13946 1/20 0.35
PDE3A Q14432 1/20 0.35
USP2 O75604 1/20 0.34
MAPT P10636 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
FFAR1 O14842 2/20 0.34
TBXA2R P21731 6/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748446 0.89 PTGDR2 (0.45) ARPPARDPPARAPDE4BCHRM1
SCHEMBL19622210 0.84 PDE4B (0.44) ARPDE4BCHRM1PDE4AADRA1A
SCHEMBL14748461 0.84 TBXA2R (0.36) ARPPARDPPARAPDE4BCHRM1
SCHEMBL14748449 0.79 PDE4B (0.38) ARPDE4BCHRM1PDE4AADRA1A
SCHEMBL8005546 0.79 AR (0.59) ARPPARDPPARAPDE4BCHRM1
SCHEMBL14748365 0.76 CYP11B1 (0.49) ARFFAR1SCN9A
SCHEMBL14748470 0.76 PDE4B (0.40) ARPDE4BCHRM1PDE4AADRA1A
SCHEMBL8005549 0.76 AR (0.44) ARPDE4BCHRM1PDE4AADRA1A
SCHEMBL14470676 0.75 PDE4B (0.53) PDE4BCHRM1PDE4AADRA1APDE1A
SCHEMBL7997146 0.74 PTGDR2 (0.42) PPARDPPARAPTGDR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed