SCHEMBL19623348

SCHEMBL19623348

NC1=NC=C(c2nc(N3CCOCC3)nc3c2CCN3)CN1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.37
PIK3R1 P27986 14/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CB P42338 1/20 0.37
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13872584 0.77 PIK3CA (0.58) PIK3CAPIK3R1PIK3CDPIK3CB
SCHEMBL2378615 0.74 PIK3CA (0.60) PIK3CAPIK3R1ALDH1A1LMNA
SCHEMBL19623320 0.72 KMT2A (0.40) PIK3CAPIK3R1PIK3CDPIK3CBALDH1A1
SCHEMBL13012640 0.72 PIK3CA (0.49) PIK3CAPIK3R1PIK3CDPIK3CB
SCHEMBL2378251 0.70 HTR2C (0.44) PIK3CAPIK3R1ALDH1A1LMNA
SCHEMBL12247675 0.70 ALDH1A1 (0.56) PIK3CAPIK3R1PIK3CDPIK3CBALDH1A1
SCHEMBL20708218 0.69 PIK3CA (0.54) PIK3CAPIK3R1PIK3CDPIK3CB
SCHEMBL13872927 0.68 PIK3CA (0.60) PIK3CAPIK3R1
SCHEMBL16684483 0.68 PIK3CA (0.37) PIK3CAPIK3R1PIK3CDPIK3CB
SCHEMBL2376887 0.65 KDM4E (0.48) PIK3CAPIK3R1PIK3CDPIK3CBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed