SCHEMBL19623540

SCHEMBL19623540

Nc1ccc(-c2nc(N3CCOCC3)nc3c2CCC3)cc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.57
PIK3R1 P27986 8/20 0.57
MTOR P42345 3/20 0.57
KDM4E B2RXH2 2/20 0.56
ALDH1A1 P00352 2/20 0.56
HPGD P15428 1/20 0.52
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623581 0.85 PIK3CA (0.60) PIK3CAPIK3R1MTORKDM4EALDH1A1
SCHEMBL24699076 0.84 KDM4E (0.50) PIK3CAPIK3R1MTORKDM4EALDH1A1
SCHEMBL24698989 0.81 PIK3CA (0.50) PIK3CAKDM4EALDH1A1HPGDLMNA
SCHEMBL24698785 0.80 KDM4E (0.50) PIK3CAPIK3R1MTORKDM4EALDH1A1
SCHEMBL19623495 0.78 KDM4E (0.57) PIK3CAMTORKDM4EALDH1A1HPGD
SCHEMBL19623545 0.78 PIK3CA (0.62) PIK3CAMTORKDM4EALDH1A1
SCHEMBL19623372 0.76 PIK3CA (0.62) PIK3CAPIK3R1MTOR
SCHEMBL24699477 0.76 ALDH1A1 (0.47) KDM4EALDH1A1HPGDMAPTNPSR1
SCHEMBL24697795 0.76 ALDH1A1 (0.40) PIK3CAKDM4EALDH1A1HPGDLMNA
SCHEMBL19623405 0.76 PIK3CA (0.52) PIK3CAKDM4EALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed