SCHEMBL19623596

SCHEMBL19623596

COCCN(C)C(=O)c1cccc(-c2nc(N3CCOCC3)nc3c2CCC(Cc2ccncc2)=C3)c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.51
MTOR P42345 1/20 0.44
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623825 0.83 PIK3CA (0.55) PIK3CAPIK3CBPIK3CG
SCHEMBL2376638 0.82 PIK3CA (0.72) PIK3CAMTOR
SCHEMBL19623809 0.80 PIK3CA (0.52) PIK3CAPIK3CBPIK3CG
SCHEMBL2377668 0.78 PIK3CA (0.65) PIK3CAMTOR
SCHEMBL19623722 0.77 PIK3CA (0.46) PIK3CAMTORPIK3CBPIK3CG
SCHEMBL12247608 0.75 PIK3CA (0.72) PIK3CA
SCHEMBL2376748 0.73 PIK3CA (0.69) PIK3CA
SCHEMBL19623577 0.72 MTOR (0.43) PIK3CAMTORPIK3CBPIK3CG
SCHEMBL12247568 0.72 PIK3CA (0.79) PIK3CA
Trifluoroacetic Acid SCHEMBL2377793 0.71 PIK3CA (0.66) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed