SCHEMBL19623809

SCHEMBL19623809

O=C(NCCCO)c1cccc(-c2nc(N3CCOCC3)nc3c2CCC(Cc2ccncc2)=C3)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.52
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42
NAMPT P43490 2/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37
MAPK14 Q16539 1/20 0.37
KDM1A O60341 1/20 0.37
HDAC1 Q13547 1/20 0.37
PARP1 P09874 1/20 0.37
ERN1 O75460 1/20 0.36
AKR1C3 P42330 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623825 0.91 PIK3CA (0.55) PIK3CAPIK3CBPIK3CGKDM1AHDAC1
SCHEMBL2376111 0.81 PIK3CA (0.77) PIK3CA
SCHEMBL19623596 0.80 PIK3CA (0.51) PIK3CAPIK3CBPIK3CG
SCHEMBL19623703 0.79 PIK3CA (0.49) PIK3CAPIK3CGNAMPTALDH1A1MAPK8
SCHEMBL19623722 0.79 PIK3CA (0.46) PIK3CAPIK3CBPIK3CG
SCHEMBL19623791 0.78 SMN1; SMN2 (0.54) PIK3CAALDH1A1MAPK8MAPK10MAPK14
SCHEMBL2379928 0.76 PIK3CA (0.67) PIK3CA
SCHEMBL2376373 0.75 PIK3CA (0.78) PIK3CA
SCHEMBL3832685 0.74 PIK3CA (0.75) PIK3CA
SCHEMBL2377284 0.73 PIK3CA (0.79) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed