SCHEMBL19623649

SCHEMBL19623649

O=C(c1cccc(-c2nc(N3CCOCC3)nc3c2CCC(Cc2cccnc2)=C3)c1)N1CCC(O)C1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 4/20 0.43
PIK3CA P42336 9/20 0.42
MTOR P42345 3/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
ROCK2 O75116 2/20 0.39
NAMPT P43490 1/20 0.37
ADORA2B P29275 1/20 0.37
ATR Q13535 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623722 0.88 PIK3CA (0.46) PIK3CAMTORPIK3CBPIK3CG
SCHEMBL12247578 0.80 PIK3CA (0.67) PIK3CA
Trifluoroacetic Acid SCHEMBL2375870 0.76 PIK3CA (0.61) PIK3CA
SCHEMBL12247595 0.76 PIK3CA (0.65) PIK3CAMTOR
SCHEMBL3835911 0.76 PIK3CA (0.72) PIK3CA
SCHEMBL2377725 0.76 PIK3CA (0.70) PIK3CA
SCHEMBL19623825 0.75 PIK3CA (0.55) PIK3CAPIK3CBPIK3CGROCK2
SCHEMBL19623646 0.73 MTOR (0.48) PIK3CAMTORPIK3CBPIK3CGATR
SCHEMBL19623809 0.72 PIK3CA (0.52) PIK3CAPIK3CBPIK3CGNAMPT
Trifluoroacetic Acid SCHEMBL2376933 0.72 PIK3CA (0.59) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed