SCHEMBL19623668

SCHEMBL19623668

CN(CCCN1CCOCC1)c1ccc(CCc2c(N)nc(N3CCOCC3)nc2-c2cnc(N)nc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.46
PIK3CD O00329 3/20 0.42
PIK3R1 P27986 12/20 0.42
MTOR P42345 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2376610 0.75 PIK3CA (0.69) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL19611202 0.73 PIK3CA (0.54) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL19623563 0.73 PIK3CA (0.55) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL2818215 0.72 PIK3CA (0.59) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL12248080 0.72 PIK3CA (0.64) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL2376765 0.72 PIK3CA (0.67) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL2377619 0.71 PIK3CA (0.70) PIK3CAPIK3CDPIK3R1MTOR
SCHEMBL19611250 0.70 PIK3CA (0.52) PIK3CAPIK3R1
SCHEMBL2375987 0.70 HTR7 (0.42)
SCHEMBL19611160 0.68 PIK3CA (0.54) PIK3CAPIK3CDPIK3R1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed