SCHEMBL19623719

SCHEMBL19623719

Cc1cccc(-c2nc(C)nc3c2CCC3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.47
MAPT P10636 4/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
HTT P42858 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
ACHE P22303 6/20 0.42
HTR7 P34969 2/20 0.42
HPGD P15428 2/20 0.41
KDM4E B2RXH2 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639510 0.81 HTR2A (0.50) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL19623475 0.80 ACHE (0.51) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL14731022 0.80 MAPT (0.42) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL19623881 0.78 HTR2A (0.38) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL14731120 0.77 MAPT (0.44) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL19623495 0.77 KDM4E (0.57) NPSR1MAPTNPC1RAB9AL3MBTL1
SCHEMBL24725927 0.77 MAPT (0.47) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL14731124 0.76 MAPT (0.43) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL16682856 0.74 MAPT (0.45) NPSR1MAPTNPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL16669168 0.72 MAPT (0.44) NPSR1MAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed