SCHEMBL19623720

SCHEMBL19623720

C=C(c1ccc(NC(C)=O)cc1)N1CCc2c(-c3cccc(O)c3)nc(N3CCOCC3)nc21

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.55
PIK3R1 P27986 4/20 0.51
MTOR P42345 2/20 0.46
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2377056 0.92 PIK3CA (0.56) PIK3CAPIK3R1MTORGAAMAPT
SCHEMBL2377364 0.84 PIK3CA (0.63) PIK3CAPIK3R1MTOR
SCHEMBL2377693 0.83 PIK3CA (0.67) PIK3CAPIK3R1MTOR
SCHEMBL2376634 0.82 PIK3CA (0.73) PIK3CAPIK3R1
SCHEMBL3224544 0.81 PIK3CA (0.71) PIK3CAPIK3R1MTOR
SCHEMBL2377490 0.81 PIK3CA (0.61) PIK3CAPIK3R1MTOR
SCHEMBL19623429 0.80 PIK3CA (0.58) PIK3CAPIK3R1
SCHEMBL27760031 0.80 PIK3CA (0.67) PIK3CAPIK3R1MTOR
SCHEMBL2378462 0.80 PIK3CA (0.60) PIK3CAPIK3R1
SCHEMBL2376941 0.79 PIK3CA (0.64) PIK3CAPIK3R1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed