SCHEMBL19623735

SCHEMBL19623735

c1cc(-c2nc(N3CCCCC3)nc3c2CCN3)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.44
L3MBTL1 Q9Y468 3/20 0.42
LMNA P02545 3/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CASP1 P29466 1/20 0.39
CASP4 P49662 1/20 0.39
CASP5 P51878 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
USP2 O75604 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
CHKA P35790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2378615 0.87 PIK3CA (0.60) PIK3CALMNAALDH1A1MAPT
SCHEMBL19623360 0.78 PIK3CA (0.46) PIK3CAL3MBTL1LMNAHPGDALDH1A1
SCHEMBL24698856 0.73 PIK3CA (0.47) PIK3CAL3MBTL1LMNAHPGDALDH1A1
SCHEMBL19623647 0.70 PIK3CA (0.50) PIK3CAL3MBTL1LMNAHPGDALDH1A1
SCHEMBL13872584 0.69 PIK3CA (0.58) PIK3CA
SCHEMBL13012640 0.69 PIK3CA (0.49) PIK3CA
SCHEMBL19623552 0.69 PIK3CA (0.69) PIK3CA
SCHEMBL2339520 0.68 HTR2C (0.61) L3MBTL1LMNAKDM4EKMT2ATDP1
SCHEMBL2339714 0.68 HTR2C (0.58) TDP1USP2SMN1; SMN2
SCHEMBL2342040 0.67 HTR2A (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed