SCHEMBL19623901

SCHEMBL19623901

CC(C)(C)Cc1cccc(-c2nc(N3CCOCC3)nc3c2CCN3)c1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.45
MTOR P42345 1/20 0.40
AOC3 Q16853 1/20 0.39
PIK3R1 P27986 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2377918 0.82 PIK3CA (0.51) PIK3CAMTOR
SCHEMBL2378615 0.76 PIK3CA (0.60) PIK3CAMTORPIK3R1
SCHEMBL13012640 0.74 PIK3CA (0.49) PIK3CAMTORPIK3R1
SCHEMBL13872584 0.72 PIK3CA (0.58) PIK3CAMTORPIK3R1
SCHEMBL12247675 0.68 ALDH1A1 (0.56) PIK3CAMTORPIK3R1
SCHEMBL24698176 0.67 KDM4E (0.44) PIK3CA
SCHEMBL10190881 0.67 AGXT (0.60)
SCHEMBL12346384 0.67 PSMB8 (0.48)
SCHEMBL2376372 0.66 PIK3CA (0.61) PIK3CAMTORPIK3R1
SCHEMBL2378251 0.66 HTR2C (0.44) PIK3CAMTORPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed