SCHEMBL19626296

SCHEMBL19626296

Cn1cc(-c2cnn(COCC[Si](C)(C)C)c2)c2cc(C#CC(C)(C)O)ccc21

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHUK O15111 14/20 0.40
MAP3K14 Q99558 4/20 0.35
TTBK1 Q5TCY1 1/20 0.34
PIKFYVE Q9Y2I7 1/20 0.32
CREBBP Q92793 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19626295 0.91 CHUK (0.46) CHUKMAP3K14TTBK1
SCHEMBL19626288 0.91 CHUK (0.48) CHUKMAP3K14PIKFYVE
SCHEMBL19626294 0.90 CHUK (0.44) CHUKMAP3K14
SCHEMBL19626292 0.90 CHUK (0.44) CHUKMAP3K14PIKFYVE
SCHEMBL19626291 0.89 CHUK (0.43) CHUKMAP3K14TTBK1PIKFYVE
SCHEMBL19629483 0.89 CHUK (0.40) CHUKMAP3K14TTBK1PIKFYVECREBBP
SCHEMBL16608293 0.86 CHUK (0.58) CHUKMAP3K14
SCHEMBL19626287 0.85 CHUK (0.50) CHUKMAP3K14CREBBP
SCHEMBL19626285 0.84 L3MBTL1 (0.36) CHUKMAP3K14
SCHEMBL19626290 0.83 CHUK (0.52) CHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9981962-B2 Pyrazole derivatives as NIK inhibitors JANSSEN PHARMACEUTICA NV (BE) 2018-05-29 US disclosed
US-9981962-B2 Pyrazole derivatives as NIK inhibitors JANSSEN PHARMACEUTICA NV (BE) 2018-05-29 US disclosed
US-20170334900-A1 NEW PYRAZOLE DERIVATIVES AS NIK INHIBITORS ARGENTA DISCOVERY 2009 LIMITED (GB) 2017-11-23 US disclosed
US-20170334900-A1 NEW PYRAZOLE DERIVATIVES AS NIK INHIBITORS ARGENTA DISCOVERY 2009 LIMITED (GB) 2017-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170334900-A1 NEW PYRAZOLE DERIVATIVES AS NIK INHIBITORS MAP3K14, MAP3K15, MAP3K21 CHUK 32/4885MAP3K14 1/4885TTBK1 713/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.