SCHEMBL19630998

SCHEMBL19630998

CCN(CC)C(=O)Oc1c(C)cc(Cl)cc1C(=O)Nc1nc2ccc(C(F)(F)F)cc2s1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 14/20 0.50
DYRK1A Q13627 1/20 0.50
ACP1 P24666 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
NCS1 P62166 1/20 0.45
CYP2D6 P10635 1/20 0.44
LRRK2 Q5S007 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631005 0.87 CSNK1D (0.55) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19612122 0.86 DYRK1A (0.57) CSNK1DDYRK1AACP1NCS1CYP2D6
SCHEMBL24044916 0.84 DYRK1A (0.54) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19612108 0.84 DYRK1A (0.54) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19612156 0.83 CSNK1D (0.50) CSNK1DDYRK1AACP1NCS1CYP2D6
SCHEMBL19612166 0.83 DYRK1A (0.53) CSNK1DDYRK1AACP1NCS1CYP2D6
SCHEMBL19612165 0.83 DYRK1A (0.53) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19627267 0.83 DYRK1A (0.53) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19630876 0.82 DYRK1A (0.51) CSNK1DDYRK1AACP1CASP3SENP8
SCHEMBL19627268 0.81 DYRK1A (0.48) CSNK1DDYRK1AACP1CASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017201313-A1 NOVEL MITOCHONDRIAL UNCOUPLERS FOR TREATMENT OF METABOLIC DISEASES AND CANCER JIN SHENGKAN (US) 2017-11-23 WO disclosed