SCHEMBL196310

SCHEMBL196310

Cc1ccc(Nc2cc(NC(=O)C3CCCCC3)c3ccccc3n2)cc1.O=C(Nc1cc(Nc2ccc(Cl)c(Cl)c2)nc2ccccc12)C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 3/20 0.47
GRM4 Q14833 1/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
TP53 P04637 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ADORA3 P0DMS8 6/20 0.44
TMEM97 Q5BJF2 3/20 0.44
SIGMAR1 Q99720 2/20 0.44
DRD3 P35462 2/20 0.44
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30637139 0.94 GRM4 (0.51) RXFP1GRM4GAAMAPTTP53
SCHEMBL29501836 0.94 GRM4 (0.51) RXFP1GRM4GAAMAPTTP53
SCHEMBL196780 0.94 GRM4 (0.51) RXFP1GRM4GAAMAPTTP53
SCHEMBL196377 0.93 GRM4 (0.49) RXFP1GRM4GAAMAPTTP53
SCHEMBL1976142 0.92 RXFP1 (0.53) RXFP1GAAMAPTTP53NPC1
SCHEMBL196452 0.91 GRM4 (0.47) RXFP1GRM4MAPTTP53NPC1
SCHEMBL935627 0.91 RXFP1 (0.51) RXFP1GAAMAPTTP53NPC1
SCHEMBL197113 0.89 MAPT (0.57) GRM4MAPTTP53RAB9AADORA3
SCHEMBL959149 0.86 RXFP1 (0.53) RXFP1GAAMAPTTP53NPC1
SCHEMBL196681 0.85 RXFP1 (0.53) RXFP1GRM4GAAMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500255-A 2012-01-05 JP claimed
EP-2323661-A1 A3 ADENOSINE RECEPTOR ALLOSTERIC MODULATORS Universiteit Leiden (NL) 2011-05-25 EP claimed
WO-2010020981-A1 A3 ADENOSINE RECEPTOR ALLOSTERIC MODULATORS UNIVERSITEIT LEIDEN (NL) 2010-02-25 WO claimed