SCHEMBL19632913

SCHEMBL19632913

C=CC1(F)CC1Cc1nnc2c(Br)c(N3CCC(c4ccccc4C)CC3)ccn12

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.44
HTR2A P28223 2/20 0.44
SLC6A3 Q01959 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633060 0.90 GRM2 (0.47) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL21084285 0.78 GRM2 (0.51) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL20842383 0.78 GRM2 (0.47) GRM2SLC6A3CYP2C9CYP2C19SIGMAR1
SCHEMBL19632915 0.71 GRM2 (0.48) GRM2SLC6A3CYP2C9CYP2C19SIGMAR1
SCHEMBL20842355 0.70 GRM2 (0.50) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL19632911 0.70 GRM2 (0.52) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL749628 0.69 GRM2 (0.77) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL19632597 0.68 GRM2 (0.52) GRM2SLC6A3CYP2C9CYP2C19SIGMAR1
SCHEMBL19633226 0.68 GRM2 (0.52) GRM2HTR2ASLC6A3CYP2C9CYP2C19
SCHEMBL19633195 0.66 GRM2 (0.62) GRM2HTR2ASLC6A3CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198180-A1 FLUORINE-CONTAINING TRIAZOLOPYRIDINE, AND MANUFACTURING METHOD, PHARMACEUTICAL COMPOSITION, AND APPLICATION THEREOF 中国科学院上海药物研究所 2017-11-23 WO disclosed