SCHEMBL19633717

SCHEMBL19633717

Brc1cccc(Nc2ccnc3cc(Br)ccc23)c1

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 3/20 0.81
EGFR P00533 10/20 0.78
GAK O14976 2/20 0.67
FADS1 O60427 1/20 0.54
PKMYT1 Q99640 1/20 0.52
FBP1 P09467 1/20 0.50
RET P07949 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633642 0.89 EGFR (0.71) ALKEGFRGAKFADS1PKMYT1
SCHEMBL19633716 0.89 ALK (0.72) ALKEGFRGAKFADS1PKMYT1
SCHEMBL19633659 0.89 ALK (0.72) ALKEGFRGAKFADS1PKMYT1
SCHEMBL4738872 0.88 EGFR (1.00) ALKEGFRGAKFADS1
SCHEMBL19633634 0.85 EGFR (0.72) ALKEGFRGAK
SCHEMBL28845712 0.85 EGFR (0.66) ALKEGFRGAKFADS1
SCHEMBL19633677 0.85 ALK (0.67) ALKEGFRGAKRET
SCHEMBL7618830 0.84 EGFR (0.68) ALKEGFRGAKFADS1PKMYT1
SCHEMBL19633704 0.83 PTK6 (0.66) ALKEGFRGAK
SCHEMBL19633507 0.81 EGFR (0.60) ALKEGFRGAKFBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed