SCHEMBL19633716

SCHEMBL19633716

Fc1cccc(Nc2ccnc3cc(Br)ccc23)c1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 5/20 0.72
EGFR P00533 4/20 0.63
GAK O14976 3/20 0.55
FADS1 O60427 1/20 0.49
TGFBR1 P36897 2/20 0.48
MAP4K4 O95819 1/20 0.48
PKMYT1 Q99640 1/20 0.48
KDR P35968 1/20 0.47
RET P07949 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633642 0.89 EGFR (0.71) ALKEGFRGAKFADS1TGFBR1
SCHEMBL19633640 0.89 GAK (0.60) ALKEGFRGAKFADS1TGFBR1
SCHEMBL19633717 0.89 ALK (0.81) ALKEGFRGAKFADS1PKMYT1
SCHEMBL19633680 0.84 FADS1 (0.63) GAKFADS1
SCHEMBL31167325 0.84 PKMYT1 (0.60) ALKEGFRGAKFADS1TGFBR1
SCHEMBL19633659 0.84 ALK (0.72) ALKEGFRGAKFADS1PKMYT1
SCHEMBL19633677 0.81 ALK (0.67) ALKEGFRGAKKDRRET
SCHEMBL19633632 0.81 GAK (0.62) EGFRGAKTGFBR1
SCHEMBL17075805 0.79 EGFR (0.74) EGFRGAK
SCHEMBL19633636 0.79 FBP1 (0.51) ALKEGFRGAKFADS1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed