SCHEMBL19634066

SCHEMBL19634066

CC(N)c1cc(Cl)ccc1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.61
HTT P42858 2/20 0.61
TP53 P04637 1/20 0.61
ADRB2 P07550 1/20 0.46
PDE2A O00408 1/20 0.44
PSEN1 P49768 3/20 0.41
PSEN2 P49810 3/20 0.41
APH1B Q8WW43 3/20 0.41
NCSTN Q92542 3/20 0.41
APH1A Q96BI3 3/20 0.41
PSENEN Q9NZ42 3/20 0.41
PNMT P11086 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
NFKB1 P19838 1/20 0.41
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
CNR1 P21554 1/20 0.38
SLC6A3 Q01959 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19627773 1.00 LMNA (0.61) LMNAHTTTP53ADRB2PDE2A
SCHEMBL20238511 1.00 LMNA (0.61) LMNAHTTTP53ADRB2PDE2A
Hydrochloric Acid SCHEMBL19613457 0.98 LMNA (0.59) LMNAHTTTP53ADRB2PDE2A
Hydrochloric Acid SCHEMBL20238264 0.98 LMNA (0.59) LMNAHTTTP53ADRB2PDE2A
Hydrochloric Acid SCHEMBL19613461 0.98 LMNA (0.59) LMNAHTTTP53ADRB2PDE2A
SCHEMBL8284264 0.85 LMNA (0.64) LMNAHTTTP53ADRB2PDE2A
SCHEMBL16046022 0.85 LMNA (0.64) LMNAHTTTP53ADRB2PDE2A
SCHEMBL13778123 0.85 LMNA (0.64) LMNAHTTTP53ADRB2PDE2A
Hydrochloric Acid SCHEMBL20791400 0.83 LMNA (0.62) LMNAHTTTP53ADRB2PDE2A
Hydrochloric Acid SCHEMBL31561539 0.83 LMNA (0.62) LMNAHTTTP53ADRB2PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110325531-B Benzenesulfonamides and their use as therapeutic agents 泽农医药公司 2022-05-27 CN disclosed
US-11174268-B2 Benzenesulfonamide compouds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2021-11-16 US disclosed
US-20210171537-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2021-06-10 US disclosed
EP-3551626-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2019-10-16 EP disclosed
WO-2018106284-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2018-06-14 WO disclosed
US-20180162868-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2018-06-14 US disclosed
WO-2017201468-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11174268-B2 Benzenesulfonamide compouds and their use as therapeutic agents KCND2, SCN1A, CACNA1D LMNA 1478/4885HTT 307/4885TP53 1710/4885
US-20210171537-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN1B, SCN2B LMNA 1080/4885HTT 509/4885TP53 1416/4885
US-20180162868-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN1B, SCN2B LMNA 1080/4885HTT 509/4885TP53 1416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.