SCHEMBL19634447

SCHEMBL19634447

CNC(=O)CNC(=O)c1ccc(CNC(C)=O)cc1

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.64
HDAC6 Q9UBN7 4/20 0.64
KMT2A Q03164 1/20 0.58
HDAC2 Q92769 6/20 0.55
HDAC3 O15379 6/20 0.55
ALDH1A1 P00352 1/20 0.54
POLB P06746 1/20 0.54
MAPT P10636 1/20 0.54
RAB9A P51151 1/20 0.54
EPHX2 P34913 5/20 0.54
NR1H4 Q96RI1 4/20 0.54
HDAC8 Q9BY41 6/20 0.51
HDAC11 Q96DB2 2/20 0.51
HDAC4 P56524 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25686649 0.85 EPHX2 (0.71) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL12368437 0.85 HDAC1 (0.74) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL21015484 0.84 HDAC6 (0.67) HDAC1HDAC6KMT2AHDAC3RAB9A
SCHEMBL19634413 0.84 NR1H4 (0.50) HDAC1HDAC6KMT2AHDAC3ALDH1A1
SCHEMBL5945692 0.84 EPHX2 (0.59) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL20180570 0.84 EPHX2 (0.50) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL19634443 0.83 HDAC1 (0.66) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL19634824 0.82 HTT (0.52) HDAC1HDAC6KMT2AHDAC2HDAC3
SCHEMBL13993336 0.82 EPHX2 (0.54) HDAC1HDAC6KMT2AMAPTEPHX2
SCHEMBL12368427 0.80 HDAC1 (0.72) HDAC1HDAC6KMT2AHDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed