SCHEMBL19634413

SCHEMBL19634413

CNC(=O)CNC(=O)c1ccc(CNC(=O)C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.50
EPHX2 P34913 4/20 0.50
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ERCC1 P07992 1/20 0.49
ERCC4 Q92889 1/20 0.49
HDAC1 Q13547 4/20 0.48
HDAC6 Q9UBN7 3/20 0.48
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
TAOK1 Q7L7X3 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22060070 0.86 NR1H4 (0.60) NR1H4EPHX2RAB9ASMN1; SMN2MEN1
SCHEMBL19634447 0.84 HDAC1 (0.64) NR1H4EPHX2RAB9AKMT2AHDAC1
SCHEMBL19634407 0.83 RAB9A (0.52) NR1H4EPHX2RAB9ASMN1; SMN2MEN1
SCHEMBL19634421 0.82 ERCC1 (0.54) NR1H4EPHX2RAB9ASMN1; SMN2MEN1
SCHEMBL20180570 0.80 EPHX2 (0.50) NR1H4EPHX2MEN1KMT2AHDAC1
SCHEMBL21015484 0.80 HDAC6 (0.67) NR1H4EPHX2RAB9AMEN1KMT2A
SCHEMBL12131750 0.79 ERCC1 (0.70) MEN1KMT2AERCC1ERCC4HDAC1
SCHEMBL13993336 0.79 EPHX2 (0.54) NR1H4EPHX2MEN1KMT2AHDAC1
SCHEMBL24904348 0.77 RAB9A (0.55) RAB9ASMN1; SMN2MEN1KMT2AHDAC1
SCHEMBL12864477 0.77 ERCC1 (0.55) RAB9ASMN1; SMN2MEN1KMT2AERCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed