SCHEMBL19634979

SCHEMBL19634979

COCc1n[nH]c(C(=O)OC)c1Br

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.45
ALDH1A1 P00352 5/20 0.39
HSD17B10 Q99714 3/20 0.39
HCAR2 Q8TDS4 1/20 0.36
MAPK1 P28482 2/20 0.34
MEN1 O00255 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 1/20 0.31
F2 P00734 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
STAT3 P40763 1/20 0.31
HIF1A Q16665 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635117 0.83 ALDH1A1 (0.36) ALDH1A1HSD17B10MAPK1MEN1HPGD
SCHEMBL23294471 0.75 KDM4C (0.50) KDM4CALDH1A1HSD17B10MAPK1MEN1
SCHEMBL29749406 0.75 KDM4C (0.65) KDM4CALDH1A1HSD17B10HCAR2MAPK1
SCHEMBL23112514 0.72 KDM4C (0.61) KDM4CALDH1A1HSD17B10HCAR2MAPK1
SCHEMBL19635175 0.72 MAPT (0.46) ALDH1A1HSD17B10MEN1HPGDKMT2A
SCHEMBL19635469 0.72 MAPT (0.43) ALDH1A1HSD17B10MAPK1HPGDKMT2A
SCHEMBL19635451 0.70 HCAR2 (0.32) HCAR2
SCHEMBL22303621 0.70 KDM4C (0.45) KDM4CALDH1A1HSD17B10MAPK1MEN1
SCHEMBL19635421 0.70 HSD17B10 (0.42) ALDH1A1HSD17B10HPGDKMT2ALMNA
SCHEMBL11205400 0.69 KDM4C (0.47) KDM4CALDH1A1HSD17B10HCAR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed