SCHEMBL19637243

SCHEMBL19637243

COc1nc2c(c(N3CCN(C(=O)OC(C)(C)C)C(CC#N)C3)n1)CCNC2

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KRAS P01116 19/20 0.39
VHL P40337 1/20 0.36
CDK7 P50613 1/20 0.36
CCNH P51946 1/20 0.36
MNAT1 P51948 1/20 0.36
SOS1 Q07889 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19637619 0.89 PARP1 (0.37) KRASPARP1
SCHEMBL29493406 0.88 KRAS (0.39) KRASVHLCDK7CCNHMNAT1
SCHEMBL19959303 0.88 KRAS (0.39) KRASVHLCDK7CCNHMNAT1
SCHEMBL30007840 0.88 PARP1 (0.35) KRASVHLCDK7CCNHMNAT1
SCHEMBL19637840 0.88 PARP1 (0.35) KRASVHLCDK7CCNHMNAT1
SCHEMBL19617060 0.88 PARP1 (0.35) KRASVHLCDK7CCNHMNAT1
SCHEMBL19637289 0.87 KRAS (0.36) KRASVHLCDK7CCNHMNAT1
SCHEMBL21319823 0.87 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL31344907 0.87 KRAS (0.45) KRASVHLCDK7CCNHMNAT1
SCHEMBL19948062 0.87 KRAS (0.36) KRASVHLCDK7CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017201161-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2017-11-23 WO disclosed