SCHEMBL1963993

SCHEMBL1963993

O=C1CCC(N2Cc3cccc(C(=O)NC(=O)c4ccc5c(c4)OCO5)c3C2=O)C(=O)N1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 15/20 0.53
MAPK1 P28482 3/20 0.52
TSHR P16473 2/20 0.52
PKM P14618 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CSNK1A1 P48729 8/20 0.46
KMT2A Q03164 3/20 0.45
USP2 O75604 2/20 0.45
MAPT P10636 2/20 0.45
POLB P06746 1/20 0.45
APEX1 P27695 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
IKZF1 Q13422 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
IKZF2 Q9UKS7 5/20 0.43
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK10 P53779 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962233 0.88 MAPK1 (0.61) CRBNMAPK1TSHRPKMHSD17B10
SCHEMBL1963600 0.85 CRBN (0.56) CRBNCSNK1A1MAPTPOLBIKZF1
SCHEMBL1962208 0.85 CRBN (0.56) CRBNCSNK1A1MAPTPOLBIKZF1
SCHEMBL1963191 0.84 CRBN (0.57) CRBNCSNK1A1MAPTPOLBIKZF1
SCHEMBL1963599 0.84 CRBN (0.64) CRBNCSNK1A1KMT2APOLBIKZF1
SCHEMBL1961875 0.84 CRBN (0.59) CRBNCSNK1A1MAPTPOLBIKZF1
SCHEMBL1962654 0.84 CRBN (0.59) CRBNCSNK1A1MAPTPOLBIKZF1
SCHEMBL1962178 0.84 CRBN (0.59) CRBNCSNK1A1KMT2APOLBIKZF1
SCHEMBL1961984 0.84 CRBN (0.59) CRBNCSNK1A1KMT2AMAPTPOLB
SCHEMBL1962021 0.83 CRBN (0.60) CRBNCSNK1A1MAPTPOLBIKZF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SI, CYP3A5, CYP2D6 CRBN 2589/4885MAPK1 4566/4885TSHR 3814/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 CRBN 2589/4885MAPK1 4566/4885TSHR 3814/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.