SCHEMBL19643108

SCHEMBL19643108

Cc1ccccc1C(=O)Oc1cccc2c1oc1c(-c3cccc(C(=O)O)c3C)cccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.51
ESR2 Q92731 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
PTGER1 P34995 1/20 0.46
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
LMNA P02545 1/20 0.44
PKM P14618 1/20 0.41
MYC P01106 1/20 0.41
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
POLB P06746 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MCL1 Q07820 2/20 0.39
BAD Q92934 1/20 0.38
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19643109 0.87 KMT2A (0.65) ESR1ESR2KMT2AMEN1KDM4E
SCHEMBL19642796 0.76 ESR1 (0.65) ESR1ESR2KMT2AMEN1KDM4E
SCHEMBL6885269 0.75 KDM4E (0.58) ESR1ESR2KMT2AMEN1PTGER1
SCHEMBL18460967 0.74 KDM4E (0.70) ESR1ESR2KMT2AMEN1KDM4E
SCHEMBL28731362 0.72 KMT2A (0.67) ESR1ESR2KMT2AMEN1KDM4E
SCHEMBL28701128 0.72 ESR1 (0.50) ESR1ESR2KMT2AMEN1PTGER1
SCHEMBL5720757 0.71 MYC (0.65) KMT2AMEN1PTGER1KDM4EHSD17B10
SCHEMBL10949915 0.71 NR4A1 (0.47) KDM4EHSD17B10LMNAMYCALDH1A1
SCHEMBL8431592 0.71 KMT2A (0.68) ESR1ESR2KMT2AMEN1KDM4E
SCHEMBL27948132 0.70 KMT2A (0.73) ESR1ESR2KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464391-B1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS BRASKEM AMERICA INC (US) 2024-01-03 EP claimed
US-11370854-B2 Non-phthalate donor for polyolefin catalysts BRASKEM AMERICA, INC. (US) 2022-06-28 US claimed
CN-109790238-B Non-phthalate donors for polyolefin catalysts 布拉斯科美国公司 2021-12-31 CN claimed
US-20200223958-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. GRACE & CO.-CONN. (US) 2020-07-16 US claimed
US-10662267-B2 Non-phthalate donor for polyolefin catalysts W.R. GRACE & CO. -CONN. (US) 2020-05-26 US claimed
US-20190270831-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W. R. GRACE & CO. - CONN. 2019-09-05 US claimed
EP-3464391-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. Grace & Co.-Conn. (US) 2019-04-10 EP claimed
WO-2017204811-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. GRACE & CO. -CONN. (US) 2017-11-30 WO claimed
EP-3464391-B1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS BRASKEM AMERICA INC (US) 2024-01-03 EP disclosed
US-11370854-B2 Non-phthalate donor for polyolefin catalysts BRASKEM AMERICA, INC. (US) 2022-06-28 US disclosed
US-11291981-B2 Boron-based electron donors for Ziegler-Natta catalyst systems BRASKEM AMERICA, INC. (US) 2022-04-05 US disclosed
CN-109790238-B Non-phthalate donors for polyolefin catalysts 布拉斯科美国公司 2021-12-31 CN disclosed
US-20200223958-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. GRACE & CO.-CONN. (US) 2020-07-16 US disclosed
EP-3668643-A1 BORON-BASED ELECTRON DONORS FOR ZIEGLER-NATTA CATALYST SYSTEMS Braskem America, Inc. (US) 2020-06-24 EP disclosed
US-10662267-B2 Non-phthalate donor for polyolefin catalysts W.R. GRACE & CO. -CONN. (US) 2020-05-26 US disclosed
US-20190270831-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W. R. GRACE & CO. - CONN. 2019-09-05 US disclosed
EP-3464391-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. Grace & Co.-Conn. (US) 2019-04-10 EP disclosed
WO-2019036376-A1 BORON-BASED ELECTRON DONORS FOR ZIEGLER-NATTA CATALYST SYSTEMS BRASKEM AMERICA, INC. (US) 2019-02-21 WO disclosed
US-20190046965-A1 BORON-BASED ELECTRON DONORS FOR ZIEGLER-NATTA CATALYST SYSTEMS BRASKEM AMERICA, INC. 2019-02-14 US disclosed
WO-2017204811-A1 NON-PHTHALATE DONOR FOR POLYOLEFIN CATALYSTS W.R. GRACE & CO. -CONN. (US) 2017-11-30 WO disclosed