SCHEMBL19643333

SCHEMBL19643333

O=C1NCCCc2c(Br)cccc21

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 7/20 0.81
PARP11 Q9NR21 6/20 0.81
PIM1 P11309 1/20 0.64
CSNK1A1 P48729 1/20 0.64
CDK5 Q00535 1/20 0.64
ROCK1 Q13464 1/20 0.64
DYRK1A Q13627 1/20 0.64
LRRK2 Q5S007 1/20 0.64
CLK4 Q9HAZ1 1/20 0.64
DYRK1B Q9Y463 1/20 0.64
PARP1 P09874 10/20 0.56
PDPK1 O15530 1/20 0.44
ACHE P22303 1/20 0.40
HSD17B10 Q99714 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2999788 0.89 PARP10 (1.00) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL29644368 0.89 PARP10 (1.00) PARP10PARP11PIM1CSNK1A1CDK5
Toluene SCHEMBL29027038 0.80 PARP10 (0.79) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL5076461 0.79 PARP1 (0.81) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL1333810 0.78 CLK4 (1.00) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL12546313 0.78 PARP10 (0.81) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL1661783 0.74 PARP10 (0.53) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL7920173 0.74 PARP10 (0.53) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL29476168 0.74 PARP10 (0.44) PARP10PARP11PIM1CSNK1A1CDK5
SCHEMBL8650202 0.74 PARP10 (0.44) PARP10PARP11PIM1CSNK1A1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12448363-B2 Kinase inhibitors VIDYA THERAPEUTICS, INC. (US) 2025-10-21 US disclosed
EP-4558483-A1 NOVEL ISOQUINOLINONE, PYRROLOPYRIDINONE AND THIENOPYRIDINONE SULFONAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2025-05-28 EP disclosed
CN-115867346-B Kinase inhibitors GB005股份有限公司 2025-03-14 CN disclosed
CN-119546576-A Novel isoquinolinones pyrrolo-pyridones and thieno pyridone sulfonamide derivatives 豪夫迈·罗氏有限公司 2025-02-28 CN disclosed
WO-2024017856-A1 NOVEL ISOQUINOLINONE, PYRROLOPYRIDINONE AND THIENOPYRIDINONE SULFONAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2024-01-25 WO disclosed
US-20230219923-A1 KINASE INHIBITORS VIDYA THERAPEUTICS, INC. 2023-07-13 US disclosed
US-20230219923-A1 KINASE INHIBITORS VIDYA THERAPEUTICS, INC. 2023-07-13 US disclosed
US-20230219923-A1 KINASE INHIBITORS VIDYA THERAPEUTICS, INC. 2023-07-13 US disclosed
EP-4157446-A1 KINASE INHIBITORS GB002, Inc. (US) 2023-04-05 EP disclosed
CN-115867346-A Kinase inhibitors GB005股份有限公司 2023-03-28 CN disclosed
US-20220127265-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2022-04-28 US disclosed
US-20220127265-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2022-04-28 US disclosed
US-11247989-B2 Therapeutic compounds and uses thereof GENENTECH, INC. (US) 2022-02-15 US disclosed
US-11247989-B2 Therapeutic compounds and uses thereof GENENTECH, INC. (US) 2022-02-15 US disclosed
EP-3464286-B1 PYRAZOLOPYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER GENENTECH INC (US) 2021-08-18 EP disclosed
US-20190241558-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2019-08-08 US disclosed
US-20190241558-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2019-08-08 US disclosed
EP-3464286-A1 PYRAZOLOPYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER Genentech, Inc. (US) 2019-04-10 EP disclosed
WO-2017205538-A1 PYRAZOLOPYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER GENENTECH, INC. (US) 2017-11-30 WO disclosed
WO-2017205538-A1 PYRAZOLOPYRIDINE DERIVATIVES FOR THE TREATMENT OF CANCER GENENTECH, INC. (US) 2017-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12448363-B2 Kinase inhibitors BTK, ABL1, LYN PARP10 732/4885PARP11 698/4885PIM1 255/4885
US-11247989-B2 Therapeutic compounds and uses thereof EP300, HDAC1, CREBBP PARP10 99/4885PARP11 61/4885PIM1 2774/4885
US-20230219923-A1 KINASE INHIBITORS BTK, ABL1, LYN PARP10 732/4885PARP11 698/4885PIM1 255/4885
US-20190241558-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF EP300, HDAC1, CREBBP PARP10 99/4885PARP11 61/4885PIM1 2774/4885
US-20220127265-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF EP300, HDAC1, CREBBP PARP10 99/4885PARP11 61/4885PIM1 2774/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.