SCHEMBL19644803

SCHEMBL19644803

CN(C)c1nc(N)nc2c1ncn2[C@@H]1OC(COP(=O)(OCCSC(=O)C(C)(C)C)OCCSC(=O)C(C)(C)C)[C@@H](O)[C@@]1(C)F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NT5E P21589 7/20 0.40
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
ENPP1 P22413 1/20 0.34
P2RY12 Q9H244 2/20 0.33
LMNA P02545 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
P2RY1 P47900 1/20 0.33
CA5A P35218 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
POLA1 P09884 1/20 0.33
P2RY11 Q96G91 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18067110 1.00 NT5E (0.40) NT5ECA12CA1CA2CA9
SCHEMBL18061705 0.92 CA12 (0.39) NT5ECA12CA1CA2CA9
SCHEMBL21136209 0.90 CA12 (0.35) NT5ECA12CA1CA2CA9
SCHEMBL18067162 0.89 ADORA1 (0.41) NT5ECA12CA1CA2CA9
SCHEMBL21015197 0.85 HTR2C (0.32) P2RY1HTR2CHTR2B
SCHEMBL19644818 0.83 CA5A (0.47) NT5EP2RY1CA5AP2RY11
SCHEMBL20841357 0.83 HTR2C (0.31) HTR2CHTR2B
SCHEMBL19822431 0.83 NT5E (0.43) NT5EP2RY12BLMP2RY1CA5A
SCHEMBL18061636 0.82 P2RY1 (0.45) NT5ECA12CA1CA2CA9
SCHEMBL18061566 0.81 P2RY1 (0.47) NT5EENPP1P2RY12P2RY1P2RY11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9828410-B2 β-D-2′-deoxy-2′-α-fluoro-2′-β-C-substituted-2-modified-N6-substituted purine nucleotides for HCV treatment Atea Pharmaceuticals, Inc. (US) 2017-11-28 US disclosed