SCHEMBL19645657

SCHEMBL19645657

COc1cc2c(=O)n(C)cnc2cc1OC(C)=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.56
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
TNF P01375 3/20 0.52
KDM4E B2RXH2 2/20 0.48
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
TNFSF11 O14788 1/20 0.45
EGFR P00533 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23959931 1.00 HDAC6 (0.56) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL4728366 0.89 HDAC6 (0.59) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL31605145 0.82 HDAC6 (0.51) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL19645655 0.80 HDAC6 (0.51) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL4782862 0.80 HDAC6 (0.51) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL24165356 0.79 HDAC6 (0.49) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL24166144 0.78 HDAC6 (0.49) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL1550700 0.78 HDAC6 (0.64) HDAC6TNFHDAC3HDAC4HDAC1
SCHEMBL19645642 0.77 HDAC6 (0.52) HDAC6TSHRMAPK1TNFKDM4E
SCHEMBL22323913 0.77 HDAC6 (0.48) HDAC6TSHRMAPK1TNFKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9827248-B2 Therapeutic compounds and uses thereof KALA PHARMACEUTICALS, INC. (US) 2017-11-28 US disclosed