SCHEMBL1965040

SCHEMBL1965040

CC(C)Oc1ccc(-c2noc(-c3ccc4cn(C(=O)O)cc4c3)n2)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.65
MAP4K4 O95819 3/20 0.59
MINK1 Q8N4C8 3/20 0.59
S1PR3 Q99500 4/20 0.58
DYRK3 O43781 1/20 0.55
MARK3 P27448 1/20 0.55
PLK1 P53350 1/20 0.55
MAP4K5 Q9Y4K4 1/20 0.55
S1PR5 Q9H228 1/20 0.54
PRKCD Q05655 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966831 0.88 S1PR1 (0.58) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL3741047 0.84 S1PR1 (0.73) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL13045365 0.81 S1PR1 (0.64) S1PR1MAP4K4MINK1S1PR3PRKCD
SCHEMBL1965044 0.80 S1PR1 (0.66) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL3746333 0.80 MAP4K4 (0.63) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL1843853 0.79 S1PR1 (0.69) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL3741171 0.79 MAP4K4 (0.65) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL398987 0.79 S1PR1 (1.00) S1PR1MAP4K4MINK1S1PR3S1PR5
SCHEMBL403510 0.79 S1PR1 (0.78) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL400101 0.79 S1PR1 (0.78) S1PR1MAP4K4MINK1S1PR3DYRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509424-A1 NOVEL OXADIAZOLE COMPOUNDS Abbott Laboratories (US) 2012-10-17 EP disclosed
WO-2011071570-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-16 WO disclosed