SCHEMBL1965044

SCHEMBL1965044

CC(C)Oc1ccc(-c2noc(-c3ccc4c(c3)CN(C(=O)O)C4)n2)cc1Cl

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.66
S1PR3 Q99500 8/20 0.66
MAP4K4 O95819 3/20 0.60
MINK1 Q8N4C8 3/20 0.60
DYRK3 O43781 1/20 0.56
MARK3 P27448 1/20 0.56
PLK1 P53350 1/20 0.56
MAP4K5 Q9Y4K4 1/20 0.56
PRKCD Q05655 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1966833 0.88 S1PR1 (0.59) S1PR1S1PR3MAP4K4MINK1DYRK3
SCHEMBL1963144 0.86 S1PR1 (0.81) S1PR1S1PR3MAP4K4MINK1
SCHEMBL1969510 0.83 S1PR1 (0.69) S1PR1S1PR3MAP4K4MINK1
SCHEMBL2989163 0.82 S1PR1 (0.60) S1PR1S1PR3MAP4K4MINK1
SCHEMBL3741047 0.82 S1PR1 (0.73) S1PR1S1PR3MAP4K4MINK1DYRK3
SCHEMBL3057688 0.82 S1PR1 (0.71) S1PR1S1PR3MAP4K4MINK1
SCHEMBL2989389 0.81 S1PR1 (0.84) S1PR1S1PR3MAP4K4MINK1
SCHEMBL1965040 0.80 S1PR1 (0.65) S1PR1S1PR3MAP4K4MINK1DYRK3
SCHEMBL1966006 0.80 S1PR1 (0.81) S1PR1S1PR3MAP4K4MINK1PRKCD
SCHEMBL2998264 0.80 S1PR1 (0.62) S1PR1S1PR3MAP4K4MINK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509424-A1 NOVEL OXADIAZOLE COMPOUNDS Abbott Laboratories (US) 2012-10-17 EP disclosed
WO-2011071570-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-16 WO disclosed