SCHEMBL1965594

SCHEMBL1965594

COc1ccc(C(=O)N(CC2CC2)c2nnc(-c3ccc(CN4CC(C(=O)OC(=O)C5CN(Cc6ccc(-c7nnc(N(CC8CC8)C(=O)Cc8ccccc8)s7)cc6)C5)C4)cc3)s2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 15/20 0.57
S1PR3 Q99500 5/20 0.46
S1PR4 O95977 1/20 0.45
S1PR5 Q9H228 1/20 0.45
ACHE P22303 1/20 0.44
CPB1 P15086 1/20 0.43
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1965593 0.94 S1PR1 (0.65) S1PR1S1PR3S1PR4S1PR5ACHE
SCHEMBL1966443 0.88 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5ACHE
SCHEMBL2295298 0.84 S1PR1 (0.75) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1964580 0.79 S1PR1 (0.68) S1PR1S1PR3S1PR4S1PR5CPB1
SCHEMBL2301982 0.75 S1PR1 (0.52) S1PR1CPB1KDM4ENPC1ALDH1A1
SCHEMBL1964739 0.75 S1PR1 (0.83) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL2298795 0.74 S1PR1 (0.51) S1PR1CPB1KDM4ENPC1ALDH1A1
SCHEMBL1965472 0.74 S1PR1 (0.81) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1966562 0.74 S1PR1 (0.74) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1965815 0.73 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP claimed
WO-2010043377-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2010-04-22 WO claimed
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP disclosed
WO-2010043377-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2010-04-22 WO disclosed