SCHEMBL1964580

SCHEMBL1964580

CCN(C(=O)Cc1ccccc1)c1nnc(-c2ccc(CN3CC(C(=O)OC(=O)C4CN(Cc5ccc(-c6nnc(N(CC)C(=O)c7ccccc7OC)s6)cc5)C4)C3)cc2)s1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.68
S1PR3 Q99500 6/20 0.55
S1PR4 O95977 1/20 0.54
S1PR5 Q9H228 1/20 0.54
KDM4E B2RXH2 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
GAA P10253 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CPB1 P15086 1/20 0.47
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1964578 0.94 S1PR1 (0.78) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1966144 0.89 S1PR1 (0.85) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1964739 0.84 S1PR1 (0.83) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1966067 0.81 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5NPC1
SCHEMBL27838327 0.81 S1PR1 (0.72) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1964349 0.79 S1PR1 (0.84) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1965594 0.79 S1PR1 (0.57) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1966168 0.77 S1PR1 (1.00) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1966562 0.77 S1PR1 (0.74) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1489208 0.77 S1PR1 (0.80) S1PR1S1PR3S1PR4S1PR5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP disclosed
WO-2010043377-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2010-04-22 WO disclosed